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BRL 50481
CAS No. 433695-36-4
BRL 50481 ( —— )
产品货号. M19908 CAS No. 433695-36-4
BRL-50481 is a novel and selective inhibitor of PDE7 with IC50s of 0.15 12.1 62 and 490 μM for PDE7A PDE7B PDE4 and PDE3 respectively.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥405 | 有现货 |
|
| 10MG | ￥486 | 有现货 |
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| 25MG | ￥1021 | 有现货 |
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| 50MG | ￥1823 | 有现货 |
|
| 100MG | ￥3062 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称BRL 50481
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述BRL-50481 is a novel and selective inhibitor of PDE7 with IC50s of 0.15 12.1 62 and 490 μM for PDE7A PDE7B PDE4 and PDE3 respectively.
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产品描述BRL-50481 is a novel and selective inhibitor of PDE7 with IC50s of 0.15 12.1 62 and 490 μM for PDE7A PDE7B PDE4 and PDE3 respectively.
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同义词——
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通路Angiogenesis
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靶点PDE
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受体PDE7
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研究领域——
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适应症——
化学信息
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CAS Number433695-36-4
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分子量244.27
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分子式C9H12N2O4S
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纯度>98% (HPLC)
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溶解度DMSO: 100 mg/mL;Ethanol: 20 mg/mL
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SMILESCN(C)S(=O)(=O)c1cc(ccc1C)[N+]([O-])=O
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化学全称NN2-Trimethyl-5-nitro-benzenesulfonamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Safavi M et al. New methods for the discovery and synthesis of PDE7 inhibitors as new drugs for neurologicaland inflammatory disorders. Expert Opin Drug Discov. 2013 Jun;8(6):733-51.
产品手册
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